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Anaplastična limfomna receptorska tirozinska kinaza

Ljudska anaplastična limfomna kinaza u kompleksu sa krizotinibom. PDB 2xp2[1]
Dostupne strukture
2KUP, 2KUQ, 2XB7, 2XBA, 2XP2, 2YFX, 2YHV, 2YJR, 2YJS, 2YS5, 2YT2, 3AOX, 3L9P, 3LCS, 3LCT, 4ANL, 4ANQ, 4ANS, 4CCB, 4CCU, 4CD0, 4DCE, 4FNW, 4FNX, 4FNY, 4FNZ, 4FOB, 4FOC, 4FOD, 4JOA, 4MKC
Identifikatori
SimboliALK; CD246; NBLST3
Vanjski IDOMIM105590 MGI103305 HomoloGene68387 GeneCards: ALK Gene
EC broj2.7.10.1
Pregled RNK izražavanja
podaci
Ortolozi
VrstaČovekMiš
Entrez23811682
EnsemblENSG00000171094ENSMUSG00000055471
UniProtQ9UM73P97793
Ref. Sekv. (iRNK)NM_004304NM_007439
Ref. Sekv. (protein)NP_004295NP_031465
Lokacija (UCSC)Chr 2:
29.42 - 30.14 Mb
Chr 17:
71.87 - 72.6 Mb
PubMed pretraga[1][2]

Reference

  1. Cui JJ, Tran-Dubé M, Shen H, Nambu M, Kung PP, Pairish M, Jia L, Meng J, Funk L, Botrous I, McTigue M, Grodsky N, Ryan K, Padrique E, Alton G, Timofeevski S, Yamazaki S, Li Q, Zou H, Christensen J, Mroczkowski B, Bender S, Kania RS, Edwards MP (September 2011). „Structure based drug design of crizotinib (PF-02341066), a potent and selective dual inhibitor of mesenchymal-epithelial transition factor (c-MET) kinase and anaplastic lymphoma kinase (ALK)”. J. Med. Chem. 54 (18): 6342–63. DOI:10.1021/jm2007613. PMID 21812414.