5-HT1D receptor

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5-hidroksitriptaminski (serotoninski) receptor 1D
Identifikatori
SimboliHTR1D; 5-HT1D; HT1DA; HTR1DA; HTRL; RDC4
Vanjski IDOMIM182133 MGI96276 HomoloGene20240 IUPHAR: 5-HT1D GeneCards: HTR1D Gene
Pregled RNK izražavanja
podaci
Ortolozi
VrstaČovekMiš
Entrez335215552
EnsemblENSG00000179546ENSMUSG00000070687
UniProtP28221Q3ZB48
RefSeq (mRNA)NM_000864NM_008309
RefSeq (protein)NP_000855NP_032335
Lokacija (UCSC)Chr 1:
23.39 - 23.39 Mb
Chr 4:
135.7 - 135.72 Mb
PubMed pretraga[1][2]

5-HT1D receptor (5-hidroksitriptaminski (serotoninski) receptor 1D, HTR1D) je 5-HT receptor. On je kodiran istoimenim genom.[1] 5-HT1D deluje na centralni nervni sistem, i utiče na kretanje i anksioznost. On takoše indukuje vaskularnu vazokonstrikciju u mozgu.

Ligandi[uredi | uredi kod]

Agonisti[uredi | uredi kod]

2

Vidi još[uredi | uredi kod]

Literatura[uredi | uredi kod]

  1. „Entrez Gene: HTR1D 5-hydroxytryptamine (serotonin) receptor 1D”. 
  2. Glennon RA, Hong SS, Dukat M, Teitler M, Davis K (1994). „5-(Nonyloxy)tryptamine: a novel high-affinity 5-HT1D beta serotonin receptor agonist”. J. Med. Chem. 37 (18): 2828–30. DOI:10.1021/jm00044a001. PMID 8071931. 
  3. Xu, YC; Schaus, JM; Walker, C; Krushinski, J; Adham, N; Zgombick, JM; Liang, SX; Kohlman, DT i dr.. (1999). „N-Methyl-5-tert-butyltryptamine: A novel, highly potent 5-HT1D receptor agonist.”. Journal of medicinal chemistry 42 (3): 526–31. DOI:10.1021/jm9805945. PMID 9986723. 
  4. „Essential psychopharmacology: neuroscientific basis and practical applications”. 

Dodatna literatura[uredi | uredi kod]

Spoljašnje veze[uredi | uredi kod]

  • „5-HT1D. IUPHAR Database of Receptors and Ion Channels. International Union of Basic and Clinical Pharmacology. Arhivirano iz originala na datum 2012-02-22.